Molecule Details
InChIKeyJDKWHSQKDBNTNC-UHFFFAOYSA-N
Compound Name7-[[1-(3-phenylphenyl)pyrazol-3-yl]methyl]-2H-triazolo[4,5-b]pyridin-5-amine
Canonical SMILESNc1cc(Cc2ccn(-c3cccc(-c4ccccc4)c3)n2)c2nn[nH]c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.12
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08684 CYP3A4 Homo sapiens Human PF00067 8.2 IC50 ChEMBL;BindingDB
P05164 MPO Homo sapiens Human PF03098 7.1 IC50 ChEMBL;BindingDB
P07202 TPO Homo sapiens Human PF03098 PF07645 PF00084 6.2 IC50 ChEMBL;BindingDB