Molecule Details
InChIKeyJDBLJGQEXWERKN-UHFFFAOYSA-N
Compound NameN-[2-[5-chloro-2-[[1-(difluoromethyl)pyrazol-4-yl]amino]pyrimidin-4-yl]oxyphenyl]prop-2-enamide
Canonical SMILESC=CC(=O)Nc1ccccc1Oc1nc(Nc2cnn(C(F)F)c2)ncc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.45
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43318 MAP3K7 Homo sapiens Human PF07714 8.2 IC50 ChEMBL;BindingDB
Q02750 MAP2K1 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P28482 MAPK1 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB