Molecule Details
InChIKeyJCXXCZVTLZJOMA-LVICEBGESA-N
Compound Name3-(4-(2-benzoylbut-1-enyl)-1-methyl-1H-pyrrol-2-yl)-N-hydroxyacrylamide
Canonical SMILESCC/C(=C\c1cc(/C=C/C(=O)NO)n(C)c1)C(=O)c1ccccc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.66
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P56524 HDAC4 Homo sapiens Human PF12203 PF00850 6.7 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 6.7 pIC50 TTD_MultiTarget
Q92769 HDAC2 Homo sapiens Human PF00850 6.7 pIC50 TTD_MultiTarget