Molecule Details
InChIKeyJCJWCXBSDFGDSJ-UHFFFAOYSA-N
Compound Name5-(2-amino-4-pyridinyl)-N-[(2-ethoxyphenyl)methyl]-2-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
Canonical SMILESCCOc1ccccc1CNc1nc(C)nc2[nH]cc(-c3ccnc(N)c3)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13627 DYRK1A Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
Q9Y463 DYRK1B Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P50750 CDK9 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB