Molecule Details
InChIKeyJCICCACMYITOCI-UHFFFAOYSA-N
Compound Name2-Methylsulfanyl-9-propan-2-yl-5,6-dihydropyrrolo[3,2-h]quinazoline-7-carboxamide
Canonical SMILESCSc1ncc2c(n1)-c1c(c(C(N)=O)cn1C(C)C)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.28
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P33981 TTK Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB