Molecule Details
InChIKeyJCAWIMDCJRNFFT-YPCKZBKDSA-N
Canonical SMILESCCCCNC(=O)C[C@H](O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)c1ccc(Oc2ccc(C(=O)N[C@@H](C)C(=O)NCCCNc3ccnc4cc(Cl)ccc34)cc2)cc1)[C@@H](C)CC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P07339 CTSD Homo sapiens Human PF07966 PF00026 6.3 IC50 ChEMBL;BindingDB
P46925 PMII Plasmodium falciparum (isolate HB3) Pathogen PF00026 8.4 Ki ChEMBL;BindingDB