Molecule Details
InChIKeyJBUCEVSQWHDZGD-VPUSJEBWSA-N
Compound Name(2S)-6-methyl-N-[(1S)-7-oxo-1-[5-(6-pyridin-3-yl-3-pyridinyl)-1H-imidazol-2-yl]nonyl]-6-azaspiro[2.5]octane-2-carboxamide
Canonical SMILESCCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2ccc(-c3cccnc3)nc2)[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O15379 HDAC3 Homo sapiens Human PF00850 8.6 IC50 ChEMBL;BindingDB
Q13547 HDAC1 Homo sapiens Human PF00850 8.4 IC50 ChEMBL;BindingDB
Q92769 HDAC2 Homo sapiens Human PF00850 7.7 IC50 ChEMBL;BindingDB