Molecule Details
InChIKeyJBLVXSZFSLHCDT-LJQANCHMSA-N
Compound Name3-[(3R)-3-aminopyrrolidin-1-yl]-1-(1-cyclooctylpiperidin-4-yl)quinoxalin-2-one
Canonical SMILESN[C@@H]1CCN(c2nc3ccccc3n(C3CCN(C4CCCCCCC4)CC3)c2=O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.45
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5TC84 OGFRL1 Homo sapiens Human PF04664 8.4 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB