Molecule Details
InChIKeyJBJIKUXUKSADFV-UHFFFAOYSA-N
Compound Name4-[[2,4-dioxo-3-(2-phenylethyl)quinazolin-1-yl]methyl]-N-hydroxybenzamide
Canonical SMILESO=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3ccccc32)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.2
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 8.4 IC50 ChEMBL;BindingDB
Q14680 MELK Homo sapiens Human PF02149 PF00069 PF21594 6.7 IC50 ChEMBL;BindingDB
Q9BY41 HDAC8 Homo sapiens Human PF00850 6.5 IC50 ChEMBL;BindingDB