Molecule Details
InChIKeyJBFFDNABQNAJAB-UHFFFAOYSA-N
Compound Name8-bromo-2-(2-chloro-3-methoxyphenyl)-3H-[1]benzofuro[3,2-d]pyrimidin-4-one
Canonical SMILESCOc1cccc(-c2nc3c(oc4ccc(Br)cc43)c(=O)[nH]2)c1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.0
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P19784 CSNK2A2 Homo sapiens Human PF00069 6.2 IC50 ChEMBL
P67870 CSNK2B Homo sapiens Human PF01214 6.2 IC50 ChEMBL