Molecule Details
InChIKeyJAGSWKLZBKKKJP-UHFFFAOYSA-N
Compound Name2,4-Diamino-5-[3',4'-Dimethoxy-5'-(5-Carboxyl-1-Pentynyl)]benzyl Pyrimidine
Canonical SMILESCOc1cc(Cc2cnc(N)nc2N)cc(C#CCCCC(=O)O)c1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P16184 Pneumocystis carinii Pathogen PF00186 9.0 IC50 ChEMBL;BindingDB
O30463 folA Mycobacterium avium Pathogen PF00186 8.6 IC50 ChEMBL;BindingDB