Molecule Details
InChIKeyIZSLXRORDBBGDE-UHFFFAOYSA-N
Compound NameN-[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]-6-[(1-prop-2-ynylpyrrolidin-2-yl)methyl]-7,8-dihydro-5H-1,6-naphthyridin-2-amine
Canonical SMILESC#CCN1CCCC1CN1CCc2nc(Nc3ncc(F)c(-c4cc(F)c5nc(C)n(C(C)C)c5c4)n3)ccc2C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB