Molecule Details
InChIKeyIYQMUEVINAUUKH-MTFGTGMQSA-N
Compound Name(E)-N-[(2R)-1-[[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methylamino]-3-methyl-1-oxobutan-2-yl]-6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enamide
Canonical SMILESCOc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)N[C@@H](C(=O)NC[C@H]1O[C@@H](n3cnc4c(N)ncnc43)[C@H](O)[C@@H]1O)C(C)C)C(=O)OC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.03
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P20839 IMPDH1 Homo sapiens Human PF00571 PF00478 8.5 Ki ChEMBL
P48449 LSS Homo sapiens Human PF13243 PF13249 8.5 Ki BindingDB
P12268 IMPDH2 Homo sapiens Human PF00571 PF00478 7.1 Ki ChEMBL;BindingDB