Molecule Details
InChIKeyIYNMVGGOTRCWGJ-CHAGIDMDSA-N
Compound NameH-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-Trp-Boc
Canonical SMILESCCCC[C@H](NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](Cc1ccccc1)NN[C@@H](Cc1ccccc1)C(=O)NCC(=O)N[C@H](C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)O)C(=O)N[C@@H](Cc1cn(C(=O)OC(C)(C)C)c2ccccc12)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.23
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P41143 OPRD1 Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P32238 CCKAR Homo sapiens Human PF00001 PF09193 Clinical TTD_MultiTarget TTD_MultiTarget