Molecule Details
InChIKeyIYNKBLIJSWYECH-LLVKDONJSA-N
Compound NameN-[(2R)-2-amino-2-[4-[4-(2-aminoethylsulfonyl)-3-sulfamoyl-2-(2H-tetrazol-5-yl)phenyl]-1H-benzimidazol-2-yl]ethyl]-2,2,2-trifluoroacetamide
Canonical SMILESNCCS(=O)(=O)c1ccc(-c2cccc3[nH]c([C@H](N)CNC(=O)C(F)(F)F)nc23)c(-c2nn[nH]n2)c1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.94
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.3 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 8.9 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.6 IC50 BindingDB