Molecule Details
InChIKeyIYFIEJRWVMLGOG-DFYNNNJYSA-N
Compound Name5-fluoro-2-(5-fluoro-1H-pyrrolo[2,3-b]pyridin-3-yl)-N-[(2S,3S)-3-(3-methyl-1,2,4-oxadiazol-5-yl)-2-bicyclo[2.2.2]octanyl]pyrimidin-4-amine
Canonical SMILESCc1noc([C@H]2C3CCC(CC3)[C@@H]2Nc2nc(-c3c[nH]c4ncc(F)cc34)ncc2F)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.01
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 6.0 Ki ChEMBL;BindingDB
P49840 GSK3A Homo sapiens Human PF00069 6.0 Ki ChEMBL
P49841 GSK3B Homo sapiens Human PF00069 6.0 Ki ChEMBL;BindingDB