Molecule Details
InChIKeyIYEGWFIGJOHWCT-UHFFFAOYSA-N
Compound Name4-Benzoyl-1-(3-hydroxyphenyl)-5-phenyl-N-(5-sulfamoyl-1,3,4-thiadiazol-2-yl)-1H-pyrazole-3-carboxamide
Canonical SMILESNS(=O)(=O)c1nnc(NC(=O)c2nn(-c3cccc(O)c3)c(-c3ccccc3)c2C(=O)c2ccccc2)s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.02
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.0 pIC50 TTD_MultiTarget
P00918 CA2 Homo sapiens Human PF00194 6.7 IC50 ChEMBL;BindingDB
P00915 CA1 Homo sapiens Human PF00194 6.4 IC50 ChEMBL;BindingDB