Molecule Details
InChIKeyIYAVTZWBGCXXFI-OCBJUFRSSA-N
Compound Name[(1R,2R,4R)-2-(4-bromophenyl)-4-morpholin-4-ylcyclohexyl]-(3,3-diphenylazetidin-1-yl)methanone
Canonical SMILESO=C([C@@H]1CC[C@@H](N2CCOCC2)C[C@H]1c1ccc(Br)cc1)N1CC(c2ccccc2)(c2ccccc2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P42785 PRCP Homo sapiens Human PF05577 8.9 IC50 ChEMBL;BindingDB
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 6.5 IC50 ChEMBL