Molecule Details
InChIKeyIVLZUGWDYRIRPP-UHFFFAOYSA-N
Compound Name5-(5-amino-2-[[3-(difluoromethoxy)pyridin-2-yl] methyl]-7-(4-fluorophenyl)-[l, 2,4]Jtriazolo[l,5-c] pyrimidin-8-yl)-1-methyl-1,2-dihydropyridin-2-one
Canonical SMILESCn1cc(-c2c(-c3ccc(F)cc3)nc(N)n3nc(Cc4ncccc4OC(F)F)nc23)ccc1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 8.4 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 8.1 IC50 ChEMBL;BindingDB