Molecule Details
InChIKeyIUOQUUDCQSGQGZ-UHFFFAOYSA-N
Compound NameN-(3-(4-(2,3-dichlorophenyl)piperazin-1-yl)propyl)-2,6-dimethylpyrimidine-4-carboxamide Hydrochloride
Canonical SMILESCc1cc(C(=O)NCCCN2CCN(c3cccc(Cl)c3Cl)CC2)nc(C)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28223 HTR2A Homo sapiens Human PF00001 6.8 IC50 ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 6.5 IC50 ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 6.2 IC50 ChEMBL;BindingDB