Molecule Details
InChIKeyIUMYNBVENHWFJF-UHFFFAOYSA-N
Compound Nameethyl 3-[4-(2-amino-1H-benzimidazol-4-yl)-2-sulfamoyl-3-(2H-tetrazol-5-yl)phenyl]sulfonylazetidine-1-carboxylate
Canonical SMILESCCOC(=O)N1CC(S(=O)(=O)c2ccc(-c3cccc4[nH]c(N)nc34)c(-c3nn[nH]n3)c2S(N)(=O)=O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.21
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.6 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.3 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.7 IC50 BindingDB