Molecule Details
InChIKeyIUMARYQWTKVJMI-UHFFFAOYSA-N
Compound Name9-cyclopropyl-7-[5-(trifluoromethyl)-1H-pyrazol-4-yl]-3H-pyrazolo[4,3-f]quinoline
Canonical SMILESFC(F)(F)c1n[nH]cc1-c1cc(C2CC2)c2c(ccc3[nH]ncc32)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P78396 CCNA1 Homo sapiens Human PF02984 PF00134 PF16500 7.1 IC50 ChEMBL
P36888 FLT3 Homo sapiens Human PF00047 PF07714 6.4 IC50 ChEMBL;BindingDB