Molecule Details
InChIKeyIUHUKZRXWQPIFE-LJAQVGFWSA-N
Compound Name2-phenyl-N-[(1S)-1-phenylpropyl]-3-[(4-propan-2-ylpiperazin-1-yl)methyl]quinoline-4-carboxamide
Canonical SMILESCC[C@H](NC(=O)c1c(CN2CCN(C(C)C)CC2)c(-c2ccccc2)nc2ccccc12)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.0
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29371 TACR3 Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P21452 TACR2 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB