Molecule Details
InChIKeyITYXRJDDBZMFAY-UHFFFAOYSA-N
Compound Name4-Chloro-N-methyl-6-(4-methyl-1-piperazinyl)-5-(methylthio)-2-pyrimidinamine
Canonical SMILESCNc1nc(Cl)c(SC)c(N2CCN(C)CC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.32
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB21271
Drug NameMezilamine
CAS Number50335-55-2
Groups experimental
ATC Codes nan
DescriptionMezilamine is a small molecule drug. Mezilamine has a monoisotopic molecular weight of 287.1 Da.

Cross-references: BindingDB: 50021365 CHEMBL407641 ZINC: ZINC000000001729
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
DrugBank Target Actions (3)
Target Gene Target Name Action Type
P08913 ADRA2A Alpha-2A adrenergic receptor inhibitor targets
P18089 ADRA2B Alpha-2B adrenergic receptor inhibitor targets
P18825 ADRA2C Alpha-2C adrenergic receptor inhibitor targets