Molecule Details
InChIKeyITMJPTIFWLPIOL-UHFFFAOYSA-N
Compound Name2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenyl-acetamide
Canonical SMILESCC(C)N(C(=O)CN1C(=O)C(NC(=O)Nc2ccccc2)C(=O)N(c2ccccc2)c2ccccc21)c1ccccc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.45
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32239 CCKBR Homo sapiens Human PF00001 7.6 IC50 ChEMBL;BindingDB
P32238 CCKAR Homo sapiens Human PF00001 PF09193 7.3 IC50 ChEMBL;BindingDB