Molecule Details
InChIKeyITFVZKLBKASFHP-NYXMJBRJSA-M
Compound NameSodium; (R)-3-acetoxymethyl-5,5,8-trioxo-7-[1-pyridin-2-yl-meth-(Z)-ylidene]-5lambda*6*-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylate
Canonical SMILESCC(=O)OCC1=C(C(=O)[O-])N2C(=O)/C(=C/c3ccccn3)[C@H]2S(=O)(=O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P05364 ampC Enterobacter cloacae Pathogen PF00144 7.6 IC50 ChEMBL;BindingDB
Q59401 Enterobacter cloacae Pathogen PF00144 6.3 IC50 ChEMBL;BindingDB
P62593 bla Escherichia coli Pathogen PF13354 6.1 IC50 ChEMBL;BindingDB