Molecule Details
InChIKeyITDPQZHRPNERLI-UHFFFAOYSA-N
Compound NameN-[2-[4-(aminomethyl)piperidin-1-yl]-5-chlorophenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
Canonical SMILESNCC1CCN(c2ccc(Cl)cc2NC(=O)c2cnn3cccnc23)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NWZ3 IRAK4 Homo sapiens Human PF07714 7.5 IC50 ChEMBL;BindingDB
P51617 IRAK1 Homo sapiens Human PF00531 PF00069 6.2 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 6.1 IC50 ChEMBL;BindingDB