Molecule Details
InChIKeyISWNVTVWJJQFQV-UHFFFAOYSA-N
Compound Name2-[[4-(3-cyclopropyl-7-fluoro-2-methylbenzimidazol-5-yl)-5-fluoropyrimidin-2-yl]amino]-N-[2-(dimethylamino)ethyl]-7,8-dihydro-5H-1,6-naphthyridine-6-carboxamide
Canonical SMILESCc1nc2c(F)cc(-c3nc(Nc4ccc5c(n4)CCN(C(=O)NCCN(C)C)C5)ncc3F)cc2n1C1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB