Molecule Details
InChIKeyISUNUPFSUDXDKD-UHFFFAOYSA-N
Compound Name7-[4-[4-[2-(2-fluoroethoxy)phenyl]piperazin-1-yl]butoxy]-1H-quinolin-2-one
Canonical SMILESO=c1ccc2ccc(OCCCCN3CCN(c4ccccc4OCCF)CC3)cc2[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.74
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 10.2 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB