Molecule Details
InChIKeyIRQIBOAVBGKTBW-UHFFFAOYSA-N
Compound Name3-[3-Tert-butylsulfanyl-5-[(5-methyl-2-pyridinyl)methoxy]-1-[[4-(5-methyl-2-pyridinyl)phenyl]methyl]indol-2-yl]-2,2-dimethylpropanoic acid
Canonical SMILESCc1ccc(COc2ccc3c(c2)c(SC(C)(C)C)c(CC(C)(C)C(=O)O)n3Cc2ccc(-c3ccc(C)cn3)cc2)nc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08684 CYP3A4 Homo sapiens Human PF00067 8.1 IC50 ChEMBL;BindingDB
P11712 CYP2C9 Homo sapiens Human PF00067 7.9 IC50 ChEMBL;BindingDB
P20292 ALOX5AP Homo sapiens Human PF01124 7.8 IC50 ChEMBL;BindingDB