Molecule Details
InChIKeyIRIDOYGIOXFPNA-UHFFFAOYSA-N
Compound Name1-Phenyl-7-pyridin-3-yl-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinoline
Canonical SMILESc1ccc(-c2nnc3n2-c2ccc(-c4cccnc4)cc2CC3)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11511 CYP19A1 Homo sapiens Human PF00067 7.7 IC50 ChEMBL;BindingDB
P05093 CYP17A1 Homo sapiens Human PF00067 7.1 IC50 ChEMBL;BindingDB
P19099 CYP11B2 Homo sapiens Human PF00067 7.0 IC50 ChEMBL;BindingDB