Molecule Details
InChIKeyIRAGSKPXCRLVGU-UHFFFAOYSA-N
Compound Name2-fluoro-6-({2-[(5-methoxy-1-{3-[4-(propan-2-yl)piperazin-1-yl]propanoyl}-2,3-dihydro-1H-indol-6-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-4-yl}amino)benzamide
Canonical SMILESCOc1cc2c(cc1Nc1nc(Nc3cccc(F)c3C(N)=O)c3cc[nH]c3n1)N(C(=O)CCN1CCN(C(C)C)CC1)CC2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.4
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06729 CD2 Homo sapiens Human PF05790 PF07686 8.4 pIC50 TTD_MultiTarget
P08069 IGF1R Homo sapiens Human PF00757 PF07714 PF01030 8.4 IC50 ChEMBL;BindingDB