Molecule Details
InChIKeyIQUJPSZZBAYWMS-JBSWOLFVSA-N
Compound Name(E)-1-[(1S,2S,6R,14R,15S,16R,20R)-11-hydroxy-15-methoxy-5-methyl-13-oxa-5,18-diazaheptacyclo[13.5.2.12,8.01,6.02,14.016,20.012,23]tricosa-8(23),9,11,21-tetraen-18-yl]-3-(4-methylphenyl)prop-2-en-1-one
Canonical SMILESCO[C@@]12C=C[C@@]3([C@@H]4CN(C(=O)/C=C/c5ccc(C)cc5)C[C@@H]41)[C@H]1Cc4ccc(O)c5c4[C@@]3(CCN1C)[C@H]2O5
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35372 OPRM1 Homo sapiens Human PF00001 9.3 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB