Molecule Details
InChIKeyIQNLJVSLHOBMFI-PRDCUKRZSA-N
Compound Name(2S)-2-{[(4R,7S,10S,13R,16S,19S)-19-amino-16-benzyl-7-[(4-hydroxy-3-iodophenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-10-({4-[(propan-2-ylamino)methyl]phenyl}methyl)-1,2-dithia-5,8,11,14,17-pentaazacycloicosan-4-yl]formamido}-3-(naphthalen-2-yl)propanamide
Canonical SMILESCC(C)NCc1ccc(C[C@@H]2NC(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)[C@H](Cc3ccccc3)NC(=O)[C@H](N)CSSC[C@@H](C(=O)N[C@@H](Cc3ccc4ccccc4c3)C(N)=O)NC(=O)[C@H](Cc3ccc(O)c(I)c3)NC2=O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.57
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32745 SSTR3 Homo sapiens Human PF00001 6.8 IC50 BindingDB
P31391 SSTR4 Homo sapiens Human PF00001 6.5 IC50 BindingDB
P30872 SSTR1 Homo sapiens Human PF00001 6.5 IC50 BindingDB