Molecule Details
InChIKeyIPUYNPMRTDZOIS-WEIBIQTGSA-N
Compound Name(2E,4E)-2,4-dimethyl-5-(6,6,9,9-tetramethyl-4-oxo-6,7,8,9-tetrahydro-4H-benzo[g]chromen-3-yl)penta-2,4-dienoic acid
Canonical SMILESCC(=C\c1coc2cc3c(cc2c1=O)C(C)(C)CCC3(C)C)/C=C(\C)C(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P10276 RARA Homo sapiens Human PF00104 PF00105 7.8 IC50 ChEMBL;BindingDB
P10826 RARB Homo sapiens Human PF00104 PF00105 7.4 IC50 ChEMBL;BindingDB
P13631 RARG Homo sapiens Human PF00104 PF00105 7.4 IC50 ChEMBL;BindingDB