Molecule Details
InChIKeyIOYFYUOBKSQTFF-UHFFFAOYSA-N
Compound Name5-bromo-4-N-[2-(1H-imidazol-5-yl)ethyl]-2-N-[3-(morpholin-4-ylmethyl)phenyl]pyrimidine-2,4-diamine
Canonical SMILESBrc1cnc(Nc2cccc(CN3CCOCC3)c2)nc1NCCc1c[nH]cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.31
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96L34 MARK4 Homo sapiens Human PF02149 PF00069 PF00627 6.7 IC50 ChEMBL;BindingDB
Q9UEE5 STK17A Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB
P27448 MARK3 Homo sapiens Human PF02149 PF00069 PF00627 6.1 IC50 ChEMBL;BindingDB