Molecule Details
InChIKeyIOUKAQLHORTKRT-UHFFFAOYSA-N
Compound Name4-[3-[2-(6-Bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine
Canonical SMILESCc1nc2ccc(-c3cc(N)nc(N)c3)nc2n1CCOc1cccc(Br)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.31
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13627 DYRK1A Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
Q92630 DYRK2 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
P50750 CDK9 Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB