Molecule Details
InChIKeyIONKULCWHLTXDF-XPZAPRPFSA-N
Compound Name[(1S,2S,5S,6R,7R,9S,10S,18R)-6-(acetyloxymethyl)-5-benzoyloxy-18-hydroxy-2,6,10-trimethyl-16-oxo-14-pyridin-3-yl-11,15-dioxatetracyclo[8.8.0.02,7.012,17]octadeca-12(17),13-dien-9-yl] 4-cyanobenzoate
Canonical SMILESCC(=O)OC[C@@]1(C)[C@@H]2C[C@H](OC(=O)c3ccc(C#N)cc3)[C@@]3(C)Oc4cc(-c5cccnc5)oc(=O)c4[C@H](O)[C@@H]3[C@@]2(C)CC[C@@H]1OC(=O)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.21
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O75908 SOAT2 Homo sapiens Human PF03062 8.0 IC50 ChEMBL;BindingDB
P35610 SOAT1 Homo sapiens Human PF03062 6.4 IC50 ChEMBL;BindingDB