Molecule Details
InChIKeyIOBUHJRBMMLWMQ-UHFFFAOYSA-N
Compound Name5-[[4-[2-(2-Methylquinolin-5-yl)oxyethyl]piperazin-1-yl]methyl]quinazoline
Canonical SMILESCc1ccc2c(OCCN3CCN(Cc4cccc5ncncc45)CC3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.17
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB