Target not found.
Molecule Details
InChIKeyINLBUQIADGPECI-UHFFFAOYSA-N
Compound Name5-(5-acetyl-2-butoxy-3-pyridinyl)-3-ethyl-2-(1-ethyl-3-azetidinyl)-2,6-dihydro-7H-pyrazolo(4,3-d)pyrimidin-7-one
Canonical SMILESCCCCOc1ncc(C(C)=O)cc1-c1nc(O)c2nn(C3CN(CC)C3)c(CC)c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.17
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O76074 PDE5A Homo sapiens Human PF01590 PF00233 8.3 IC50 ChEMBL;BindingDB
P51160 PDE6C Homo sapiens Human PF01590 PF00233 6.1 IC50 ChEMBL