Molecule Details
InChIKeyINIAMHAOELUABG-UHFFFAOYSA-N
Compound Name3-[6-(3-Dimethylamino-phenoxy)-3,5-difluoro-4-methyl-pyridin-2-yloxy]-4-hydroxy-benzamidine
Canonical SMILESCc1c(F)c(Oc2cccc(N(C)C)c2)nc(Oc2cc(C(=N)N)ccc2O)c1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.08
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 8.5 Ki ChEMBL;BindingDB
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.7 Ki ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 6.0 Ki BindingDB