Molecule Details
InChIKeyINGBKPUFSDYYRV-UHFFFAOYSA-N
Canonical SMILESCc1nnc(N2CCCC2)c2nn(-c3ccc(Cl)cc3Cl)c(C)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P54289 CACNA2D1 Homo sapiens Human PF08473 PF00092 PF08399 7.6 IC50 ChEMBL;BindingDB
Q9NY47 CACNA2D2 Homo sapiens Human PF08473 PF00092 PF08399 6.2 IC50 ChEMBL;BindingDB