Molecule Details
InChIKeyINARDHYYJBOMKR-UHFFFAOYSA-N
Compound Name6-[1-[6-(1-Piperazinyl)-2-pyridinyl]-1H-pyrazolo[4,3-c]pyridin-6-yl]-2-pyrazinecarbonitrile
Canonical SMILESN#Cc1cncc(-c2cc3c(cn2)cnn3-c2cccc(N3CCNCC3)n2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.74
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.4 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.0 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.8 Ki ChEMBL;BindingDB