Molecule Details
InChIKeyIMARJVJNXLXPIX-UHFFFAOYSA-N
Compound Name3-[4-[[[(2-Chlorophenyl)amino]carbonyl]amino]-1H-pyrazol-1-yl]-N-[1-(3-pyrrolidinyl)-1H-pyrazol-4-yl]benzamide
Canonical SMILESO=C(Nc1cnn(-c2cccc(C(=O)Nc3cnn(C4CCNC4)c3)c2)c1)Nc1ccccc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45984 MAPK9 Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.7 IC50 ChEMBL
P45983 MAPK8 Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB