Molecule Details
InChIKeyILVKGSGRGSOAHZ-UHFFFAOYSA-N
Compound Name3-[3-[4-(aminomethyl)phenyl]-5-(1H-pyrazol-4-yl)imidazo[4,5-b]pyridin-2-yl]pyridin-2-amine
Canonical SMILESNCc1ccc(-n2c(-c3cccnc3N)nc3ccc(-c4cn[nH]c4)nc32)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31751 AKT2 Homo sapiens Human PF00169 PF00069 PF00433 7.8 IC50 ChEMBL;BindingDB
P31749 AKT1 Homo sapiens Human PF00169 PF00069 PF00433 7.8 IC50 ChEMBL;BindingDB
Q9Y243 AKT3 Homo sapiens Human PF00169 PF00069 PF00433 7.2 IC50 ChEMBL;BindingDB