Molecule Details
InChIKeyILTSJNSAHXKVSQ-FVMQRRFMSA-N
Compound Namealpha-melanotropin-II(MT-II) peptide
Canonical SMILESCCCC[C@H](NC(C)=O)C(=O)N[C@H]1CC(=O)NCCCCC[C@@H](C(N)=O)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]cn2)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.69
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB