Molecule Details
InChIKeyIKXUQDQGFGOUFF-ZETCQYMHSA-N
Compound Name3-(fluoromethyl)-1-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]-7H-pyrazolo[5,4-d]pyrimidine-4,6-dione
Canonical SMILESC[C@@H](c1ccc(C(F)(F)F)cc1)n1nc(CF)c2c(=O)[nH]c(O)nc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.1
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O00408 PDE2A Homo sapiens Human PF01590 PF00233 8.2 Ki ChEMBL;BindingDB
O76083 PDE9A Homo sapiens Human PF00233 6.0 IC50 ChEMBL;BindingDB