Molecule Details
InChIKeyIKUAJUBZHRXQPW-PTLVVNQVSA-N
Compound Name(S)-4-[3-(2-{(S)-3-[((S)-1-Phenyl-ethylamino)-methyl]-pyrrolidin-1-yl}-ethyl)-1H-indol-5-ylmethyl]-oxazolidin-2-one
Canonical SMILESC[C@H](NC[C@@H]1CCN(CCc2c[nH]c3ccc(C[C@H]4COC(=O)N4)cc23)C1)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 9.5 IC50 ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 8.1 IC50 ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 7.3 IC50 ChEMBL;BindingDB