Molecule Details
InChIKeyIKIAJUVGDUYASS-UHFFFAOYSA-N
Compound Name4-[[(6-Hydroxy-4,5,7-trimethyl-1,3-benzothiazol-2-yl)amino]methyl]benzenesulfonamide
Canonical SMILESCc1c(O)c(C)c2sc(NCc3ccc(S(N)(=O)=O)cc3)nc2c1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.08
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15722 LTB4R Homo sapiens Human PF00001 7.5 IC50 ChEMBL;BindingDB
P09917 ALOX5 Homo sapiens Human PF00305 PF01477 6.6 IC50 ChEMBL;BindingDB