Molecule Details
InChIKeyIKFMCZJWBBXODH-MJBXVCDLSA-N
Compound Name(2S,11S,12R)-11-N-hydroxy-2-N-methyl-12-(2-methylpropyl)-8,13-dioxo-1,7-diazacyclotridecane-2,11-dicarboxamide
Canonical SMILESCNC(=O)[C@@H]1CCCCNC(=O)CC[C@H](C(=O)NO)[C@@H](CC(C)C)C(=O)N1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.71
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P03956 MMP1 Homo sapiens Human PF00045 PF00413 PF01471 8.8 Ki ChEMBL;BindingDB
Q9ULZ9 MMP17 Homo sapiens Human PF00045 PF00413 PF01471 8.8 pIC50 TTD_MultiTarget
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 8.4 Ki ChEMBL;BindingDB